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- W1946345724 abstract "NMR spectroscopy is a powerful technique for determining the structures of molecules in solution. It involves placing a sample in a powerful magnetic field and irradiating it with radio waves of defined frequency. The emitted signals provide information about the local molecular environments of nuclei in the sample, from which structures can be derived. NMR can also be used for determining interactions between molecules and is particularly useful for determining the nature of binding interactions between ligands and macromolecules. This information is very important in drug design: by understanding how bioactive molecules interact with a target protein or nucleic acid it is, in principle, possible to design ligands with improved affinity and specificity, which may make useful drug leads. In addition to this structure-based approach to drug design, NMR is also useful as a screening tool in drug discovery programs to identify ligands that bind to target macromolecules." @default.
- W1946345724 created "2016-06-24" @default.
- W1946345724 creator A5033914141 @default.
- W1946345724 creator A5055317480 @default.
- W1946345724 date "2006-09-15" @default.
- W1946345724 modified "2023-09-23" @default.
- W1946345724 title "Structure-based Drug Design and NMR-based Screening" @default.
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