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- W2083413390 endingPage "213" @default.
- W2083413390 startingPage "206" @default.
- W2083413390 abstract "Overdoses of carvedilol result mainly in hypotension and bradycardia. For excessive bradycardia, atropine is used successfully, while to support ventricular function intravenous glucagon, dobutamine, or isoproterenol is recommended. For severe hypotension, adrenaline or noradrenaline can be given. Glyceryl trinitrate is used for its relaxing action on smooth muscle during cesarean delivery, with the aim of facilitating fetal extraction. Ciclosporin increases the survival of allografts in humans. However, it causes renal vasoconstriction and increases proximal tubular reabsorption, leading in some cases to hypertension. The concomitant use of calcium antagonists can prevent most of the adverse effects of ciclosporin. However, some calcium antagonists (verapamil, diltiazem, nicardipine) can increase plasma concentrations of cyclosporin up to three-fold through the inhibition of cytochrome P450. Verapamil is both a substrate and an inhibitor of CYP3A4, which is inhibited by clarithromycin and erythromycin. Giving these macrolide antibiotics during verapamil therapy reduces the first-pass metabolism of verapamil, increases its systemic availability, and impairs its elimination." @default.
- W2083413390 created "2016-06-24" @default.
- W2083413390 creator A5057872974 @default.
- W2083413390 creator A5083771783 @default.
- W2083413390 creator A5088186128 @default.
- W2083413390 date "2000-01-01" @default.
- W2083413390 modified "2023-09-27" @default.
- W2083413390 title "β-adrenoceptor antagonists and antianginal drugs" @default.
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