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- NCIT_C102875 IAO_0000115 "A formulation of nanoparticles encapsulating the hydrochloride salt form of the anthracycline antibiotic doxorubicin, with potential antitumor activity. Upon intravenous administration, doxorubicin intercalates DNA, interferes with the activity of topoisomerase II, and causes DNA adducts and other DNA damage, resulting in tumor cell growth inhibition and apoptosis. This agent also interacts with cell membrane lipids causing lipid peroxidation. Delivery of doxorubicin in nanoparticles may improve drug penetration into tumors and may circumvent the tumor cells multidrug resistance mechanisms and may therefore be effective in chemoresistant tumor cells." @default.
- NCIT_C102875 NCIT_A32 NCIT_C1909 @default.
- NCIT_C102875 NCIT_NHC0 "C102875" @default.
- NCIT_C102875 NCIT_P106 "Pharmacologic Substance" @default.
- NCIT_C102875 NCIT_P108 "Nanoparticle-encapsulated Doxorubicin Hydrochloride" @default.
- NCIT_C102875 NCIT_P208 "CL437178" @default.
- NCIT_C102875 NCIT_P322 "GDC" @default.
- NCIT_C102875 NCIT_P329 "738259" @default.
- NCIT_C102875 NCIT_P330 "738259" @default.
- NCIT_C102875 NCIT_P375 "Nanoparticle-encapsulated Doxorubicin Hydrochloride" @default.
- NCIT_C102875 NCIT_P399 "738259" @default.
- NCIT_C102875 normalizedInformationContent "100" @default.
- NCIT_C102875 referenceCount "1" @default.
- NCIT_C102875 hasExactSynonym "BA-003" @default.
- NCIT_C102875 hasExactSynonym "Doxorubicin Transdrug" @default.
- NCIT_C102875 hasExactSynonym "Livatag" @default.
- NCIT_C102875 hasExactSynonym "Nanoparticle-encapsulated Doxorubicin Hydrochloride" @default.
- NCIT_C102875 inSubset NCIT_C128784 @default.
- NCIT_C102875 inSubset NCIT_C157711 @default.
- NCIT_C102875 inSubset NCIT_C157712 @default.
- NCIT_C102875 inSubset NCIT_C176424 @default.
- NCIT_C102875 inSubset NCIT_C177537 @default.
- NCIT_C102875 type Class @default.
- NCIT_C102875 isDefinedBy ncit.owl @default.
- NCIT_C102875 label "Nanoparticle-encapsulated Doxorubicin Hydrochloride" @default.
- NCIT_C102875 subClassOf NCIT_C102875 @default.
- NCIT_C102875 subClassOf NCIT_C129824 @default.
- NCIT_C102875 subClassOf NCIT_C129825 @default.
- NCIT_C102875 subClassOf NCIT_C1594 @default.
- NCIT_C102875 subClassOf NCIT_C1748 @default.
- NCIT_C102875 subClassOf NCIT_C186664 @default.
- NCIT_C102875 subClassOf NCIT_C1908 @default.
- NCIT_C102875 subClassOf NCIT_C1909 @default.
- NCIT_C102875 subClassOf NCIT_C1968 @default.
- NCIT_C102875 subClassOf NCIT_C2115 @default.
- NCIT_C102875 subClassOf NCIT_C2161 @default.
- NCIT_C102875 subClassOf NCIT_C2189 @default.
- NCIT_C102875 subClassOf NCIT_C259 @default.
- NCIT_C102875 subClassOf NCIT_C274 @default.
- NCIT_C102875 subClassOf NCIT_C2842 @default.
- NCIT_C102875 subClassOf NCIT_C471 @default.
- NCIT_C102875 subClassOf NCIT_C67502 @default.