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- NCIT_C165655 IAO_0000115 "A small molecule analogue of cyclic GMP-AMP (cGAMP) that acts as an agonist of the stimulator of interferon genes protein (STING; transmembrane protein 173; TMEM173) with potential immunoactivating and antineoplastic activities. Upon intratumoral administration, STING agonist IMSA101 binds to STING and activates STING-mediated pathways. This activates the immune response through the activation of certain immune cells which induces the expression of pro-inflammatory cytokines and chemokines, promotes tumor-associated antigen (TAA) processing and presentation by dendritic cells (DCs) and leads to an antigen-specific T-cell mediated immune response against cancer cells. STING, a transmembrane protein that activates immune cells in the tumor microenvironment, plays a key role in the activation of the innate immune system." @default.
- NCIT_C165655 NCIT_A32 NCIT_C1909 @default.
- NCIT_C165655 NCIT_A7 NCIT_C101588 @default.
- NCIT_C165655 NCIT_NHC0 "C165655" @default.
- NCIT_C165655 NCIT_P106 "Pharmacologic Substance" @default.
- NCIT_C165655 NCIT_P107 "STING Agonist IMSA101" @default.
- NCIT_C165655 NCIT_P108 "STING Agonist IMSA101" @default.
- NCIT_C165655 NCIT_P208 "CL978957" @default.
- NCIT_C165655 NCIT_P322 "CTRP" @default.
- NCIT_C165655 NCIT_P322 "GDC" @default.
- NCIT_C165655 NCIT_P329 "800118" @default.
- NCIT_C165655 NCIT_P330 "800118" @default.
- NCIT_C165655 NCIT_P375 "STING Agonist IMSA101" @default.
- NCIT_C165655 NCIT_P399 "800118" @default.
- NCIT_C165655 normalizedInformationContent "100" @default.
- NCIT_C165655 referenceCount "1" @default.
- NCIT_C165655 hasExactSynonym "IMSA 101" @default.
- NCIT_C165655 hasExactSynonym "IMSA-101" @default.
- NCIT_C165655 hasExactSynonym "IMSA101" @default.
- NCIT_C165655 hasExactSynonym "STING Agonist IMSA101" @default.
- NCIT_C165655 inSubset NCIT_C116977 @default.
- NCIT_C165655 inSubset NCIT_C116978 @default.
- NCIT_C165655 inSubset NCIT_C128784 @default.
- NCIT_C165655 inSubset NCIT_C157711 @default.
- NCIT_C165655 inSubset NCIT_C157712 @default.
- NCIT_C165655 inSubset NCIT_C176424 @default.
- NCIT_C165655 inSubset NCIT_C177537 @default.
- NCIT_C165655 type Class @default.
- NCIT_C165655 isDefinedBy ncit.owl @default.
- NCIT_C165655 label "STING Agonist IMSA101" @default.
- NCIT_C165655 subClassOf NCIT_C129820 @default.
- NCIT_C165655 subClassOf NCIT_C165655 @default.
- NCIT_C165655 subClassOf NCIT_C176586 @default.
- NCIT_C165655 subClassOf NCIT_C1908 @default.
- NCIT_C165655 subClassOf NCIT_C1909 @default.
- NCIT_C165655 subClassOf NCIT_C274 @default.
- NCIT_C165655 subClassOf NCIT_C308 @default.