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- NCIT_C180527 IAO_0000115 "An orally bioavailable, selective, small molecule inhibitor of FMS-like tyrosine kinase 3 (FLT3; CD135; STK1; FLK2), with potential antineoplastic activity. Upon oral administration, clifutinib targets, binds to and inhibits the activity of FLT3. This inhibits the proliferation of FLT3-expressing cancer cells. FLT3, a class III receptor tyrosine kinase (RTK), is overexpressed or mutated in most B-lineage neoplasms and in acute myeloid leukemias." @default.
- NCIT_C180527 NCIT_A5 NCIT_C180526 @default.
- NCIT_C180527 NCIT_A7 NCIT_C26202 @default.
- NCIT_C180527 NCIT_NHC0 "C180527" @default.
- NCIT_C180527 NCIT_P106 "Pharmacologic Substance" @default.
- NCIT_C180527 NCIT_P108 "Clifutinib" @default.
- NCIT_C180527 NCIT_P208 "CL1663048" @default.
- NCIT_C180527 NCIT_P322 "GDC" @default.
- NCIT_C180527 normalizedInformationContent "100" @default.
- NCIT_C180527 referenceCount "1" @default.
- NCIT_C180527 hasExactSynonym "Clifutinib" @default.
- NCIT_C180527 inSubset NCIT_C128784 @default.
- NCIT_C180527 inSubset NCIT_C157711 @default.
- NCIT_C180527 inSubset NCIT_C157712 @default.
- NCIT_C180527 type Class @default.
- NCIT_C180527 isDefinedBy ncit.owl @default.
- NCIT_C180527 label "Clifutinib" @default.
- NCIT_C180527 subClassOf NCIT_C124800 @default.
- NCIT_C180527 subClassOf NCIT_C1404 @default.
- NCIT_C180527 subClassOf NCIT_C163758 @default.
- NCIT_C180527 subClassOf NCIT_C163790 @default.
- NCIT_C180527 subClassOf NCIT_C180527 @default.
- NCIT_C180527 subClassOf NCIT_C1908 @default.
- NCIT_C180527 subClassOf NCIT_C1909 @default.
- NCIT_C180527 subClassOf NCIT_C1967 @default.
- NCIT_C180527 subClassOf NCIT_C274 @default.
- NCIT_C180527 subClassOf NCIT_C471 @default.