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- NCIT_C91731 IAO_0000115 "An orally available agent targeting phosphatidylinositol 3 kinase (PI3K) and mammalian target of rapamycin (mTOR) kinase in the PI3K/mTOR signaling pathway, with potential antineoplastic activity. Apitolisib inhibits both PI3K kinase and mTOR kinase, which may result in tumor cell apoptosis and growth inhibition of cancer cells overexpressing PI3K/mTOR. Activation of the PI3K/mTOR pathway promotes cell growth, survival, and resistance to chemotherapy and radiotherapy; mTOR, a serine/threonine kinase downstream of PI3K, may also be activated in a PI3K-independent fashion." @default.
- NCIT_C91731 NCIT_A32 NCIT_C1909 @default.
- NCIT_C91731 NCIT_A7 NCIT_C17411 @default.
- NCIT_C91731 NCIT_NHC0 "C91731" @default.
- NCIT_C91731 NCIT_P106 "Pharmacologic Substance" @default.
- NCIT_C91731 NCIT_P107 "Apitolisib" @default.
- NCIT_C91731 NCIT_P108 "Apitolisib" @default.
- NCIT_C91731 NCIT_P207 "C2984520" @default.
- NCIT_C91731 NCIT_P210 "1032754-93-0" @default.
- NCIT_C91731 NCIT_P319 "1C854K1MIJ" @default.
- NCIT_C91731 NCIT_P322 "CTRP" @default.
- NCIT_C91731 NCIT_P322 "FDA" @default.
- NCIT_C91731 NCIT_P322 "GDC" @default.
- NCIT_C91731 NCIT_P329 "639518" @default.
- NCIT_C91731 NCIT_P330 "639518" @default.
- NCIT_C91731 NCIT_P375 "Apitolisib" @default.
- NCIT_C91731 NCIT_P399 "639518" @default.
- NCIT_C91731 normalizedInformationContent "100" @default.
- NCIT_C91731 referenceCount "1" @default.
- NCIT_C91731 hasExactSynonym "APITOLISIB" @default.
- NCIT_C91731 hasExactSynonym "Apitolisib" @default.
- NCIT_C91731 hasExactSynonym "GDC 0980" @default.
- NCIT_C91731 hasExactSynonym "GDC-0980" @default.
- NCIT_C91731 hasExactSynonym "GNE 390" @default.
- NCIT_C91731 hasExactSynonym "RG 7422" @default.
- NCIT_C91731 inSubset NCIT_C116977 @default.
- NCIT_C91731 inSubset NCIT_C116978 @default.
- NCIT_C91731 inSubset NCIT_C128784 @default.
- NCIT_C91731 inSubset NCIT_C157711 @default.
- NCIT_C91731 inSubset NCIT_C157712 @default.
- NCIT_C91731 inSubset NCIT_C176424 @default.
- NCIT_C91731 inSubset NCIT_C177537 @default.
- NCIT_C91731 inSubset NCIT_C63923 @default.
- NCIT_C91731 type Class @default.
- NCIT_C91731 isDefinedBy ncit.owl @default.
- NCIT_C91731 label "Apitolisib" @default.
- NCIT_C91731 subClassOf NCIT_C129824 @default.
- NCIT_C91731 subClassOf NCIT_C129825 @default.
- NCIT_C91731 subClassOf NCIT_C1404 @default.
- NCIT_C91731 subClassOf NCIT_C163758 @default.
- NCIT_C91731 subClassOf NCIT_C1742 @default.
- NCIT_C91731 subClassOf NCIT_C1908 @default.
- NCIT_C91731 subClassOf NCIT_C1909 @default.
- NCIT_C91731 subClassOf NCIT_C2152 @default.
- NCIT_C91731 subClassOf NCIT_C2189 @default.
- NCIT_C91731 subClassOf NCIT_C2201 @default.
- NCIT_C91731 subClassOf NCIT_C274 @default.
- NCIT_C91731 subClassOf NCIT_C471 @default.
- NCIT_C91731 subClassOf NCIT_C61074 @default.
- NCIT_C91731 subClassOf NCIT_C91731 @default.