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- W1009090028 abstract "Publisher Summary This chapter discusses the nitrogen mustards and related alkylating agents. Interest in the alkylating agents primarily stems from their potentialities in the chemotherapy of cancer. But two decades of endeavor in this direction have engendered, at best, only guarded optimism concerning their efficacy, and it may well be that none will find a lasting place in the pharmacopoeia. Even so, they are certainly of proved value as tools of fundamental research, and an attempt is made to demonstrate this by presenting a broad picture of some recent studies bearing on their pharmacological action. The drugs which are now customarily grouped together as “alkylating agents of the mustard type” are the nitrogen and sulfur mustards themselves, and the bis-sulfonic esters, ethyleneimines, and ethylene oxides. Such compounds can formally be regarded as having potential alkylating properties by virtue of their being precursors of difunctional carbonium." @default.
- W1009090028 created "2016-06-24" @default.
- W1009090028 creator A5055697692 @default.
- W1009090028 date "1963-01-01" @default.
- W1009090028 modified "2023-09-27" @default.
- W1009090028 title "Nitrogen Mustards and Related Alkylating Agents" @default.
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