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- W104910708 endingPage "188" @default.
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- W104910708 abstract "It has been accepted for several years that opioid action mediated through μ- and δ-type opioid receptors requires the interaction of the agonist- occupied receptor with a guanine nucleotide binding protein (G protein). Accumulating evidence suggests that a similar mechanism is an essential component of κ-type opioid receptor function. In this chapter, we will discuss the evidence supporting these conclusions and review similarities and differences between opioid receptor-G protein interactions and the functions of other G protein-linked receptor systems. The evidence that tolerance to opioid agonist actions and the development of dependence on opioid agonist after chronic exposure might also be related to modified interactions between receptor and G protein, and also to changes in the concentrations of individual forms of G proteins, will also be considered." @default.
- W104910708 created "2016-06-24" @default.
- W104910708 creator A5084186413 @default.
- W104910708 date "1993-01-01" @default.
- W104910708 modified "2023-10-03" @default.
- W104910708 title "Opioid Receptor-G Protein Interactions: Acute and Chronic Effects of Opioids" @default.
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