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- W107344 abstract "Displacement of specific 3H-dihydroergocryptine (3H-DHE) binding to brain membranes by prazosin or yohimbine give biphasic displacement curves. Dose-dependent binding of 3H-DHE in the presence of prazosin or yohimbine in excess is saturable and Scatchard plots give Kd's for ‘prazosin’ (α1) and ‘yohimbine’ (α2) sites of 4.7 nM and 3.3 nM respectively. Saturation of ‘α2’ sites permits 3H-DHE to bind to ‘α1’ sites. Prazosin, but not ‘yohimbine-like’ drugs, displaces the ligand from these sites, and conversely for blockade of ‘α1’ sites. Two types of α-receptors thus exist in brain." @default.
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- W107344 date "1979-01-01" @default.
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- W107344 title "BIOCHEMICAL EVIDENCE FOR ‘PRE-’ AND ‘POSTSYNAPTIC’ ALPHA ADRENOCEPTORS IN RAT BRAIN" @default.
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- W107344 doi "https://doi.org/10.1016/b978-1-4832-8363-0.50175-0" @default.
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