Matches in SemOpenAlex for { <https://semopenalex.org/work/W115174184> ?p ?o ?g. }
- W115174184 abstract "Membrane transporters belong to two major super families, ATP binding cassette (ABC) transporters and solute carriers (SLC), and play a central role in body homeostasis regulation. Among these membrane proteins, the transporters carrying drugs are extensively studied and participate into the protection of the body against xenobiotics. Drug transporters are involved in all aspects of drugs absorption, disposition, and excretion. Several ABC transporters are highly overexpressed in various tumors and play an important role in the development of multidrug resistance phenotypes in cancers. Furthermore, several transporter polymorphisms have been shown to alter the pharmacokinetic profile of drugs in clinics. Drug transporters are, therefore, biomarkers of drug pharmacodynamics and pharmacokinetics. Finally, transporter substrates can also serve as biomarkers when transporter function is impaired. This chapter reviews the recent research progress in this field with an emphasis on the use of drug transporters as biomarkers in clinics." @default.
- W115174184 created "2016-06-24" @default.
- W115174184 creator A5075831790 @default.
- W115174184 creator A5080845131 @default.
- W115174184 creator A5054368831 @default.
- W115174184 date "2014-01-01" @default.
- W115174184 modified "2023-10-08" @default.
- W115174184 title "Membrane transporters and transporter substrates as biomarkers for drug pharmacokinetics, pharmacodynamics, and toxicity/adverse events" @default.
- W115174184 cites W104199933 @default.
- W115174184 cites W1550300650 @default.
- W115174184 cites W1553284301 @default.
- W115174184 cites W1567907251 @default.
- W115174184 cites W1571331723 @default.
- W115174184 cites W1598432003 @default.
- W115174184 cites W1754555893 @default.
- W115174184 cites W1807625460 @default.
- W115174184 cites W1828787736 @default.
- W115174184 cites W1888080914 @default.
- W115174184 cites W1964724251 @default.
- W115174184 cites W1966580925 @default.
- W115174184 cites W1966859174 @default.
- W115174184 cites W1968067958 @default.
- W115174184 cites W1968145453 @default.
- W115174184 cites W1969405789 @default.
- W115174184 cites W1972016245 @default.
- W115174184 cites W1972152785 @default.
- W115174184 cites W1974529503 @default.
- W115174184 cites W1975155494 @default.
- W115174184 cites W1977668920 @default.
- W115174184 cites W1979496764 @default.
- W115174184 cites W1979613025 @default.
- W115174184 cites W1980916618 @default.
- W115174184 cites W1981016777 @default.
- W115174184 cites W1981814969 @default.
- W115174184 cites W1985531970 @default.
- W115174184 cites W1985773018 @default.
- W115174184 cites W1986885996 @default.
- W115174184 cites W1987598198 @default.
- W115174184 cites W1987674565 @default.
- W115174184 cites W1989061195 @default.
- W115174184 cites W1990706522 @default.
- W115174184 cites W1991498477 @default.
- W115174184 cites W1991953785 @default.
- W115174184 cites W1992309965 @default.
- W115174184 cites W1993088391 @default.
- W115174184 cites W1993494709 @default.
- W115174184 cites W1994484433 @default.
- W115174184 cites W1995050403 @default.
- W115174184 cites W1995408306 @default.
- W115174184 cites W1995975317 @default.
- W115174184 cites W1996583648 @default.
- W115174184 cites W1997003352 @default.
- W115174184 cites W1997038641 @default.
- W115174184 cites W1997486990 @default.
- W115174184 cites W1997539457 @default.
- W115174184 cites W1997730952 @default.
- W115174184 cites W1998782146 @default.
- W115174184 cites W1999659639 @default.
- W115174184 cites W1999792279 @default.
- W115174184 cites W2000273540 @default.
- W115174184 cites W2000484916 @default.
- W115174184 cites W2000710902 @default.
- W115174184 cites W2002038028 @default.
- W115174184 cites W2002253438 @default.
- W115174184 cites W2004550238 @default.
- W115174184 cites W2005615400 @default.
- W115174184 cites W2005727737 @default.
- W115174184 cites W2010488171 @default.
- W115174184 cites W2012153991 @default.
- W115174184 cites W2014283537 @default.
- W115174184 cites W2014565106 @default.
- W115174184 cites W2016562008 @default.
- W115174184 cites W2018258967 @default.
- W115174184 cites W2021677985 @default.
- W115174184 cites W2023154099 @default.
- W115174184 cites W2023434765 @default.
- W115174184 cites W2023939814 @default.
- W115174184 cites W2024937262 @default.
- W115174184 cites W2025760569 @default.
- W115174184 cites W2026399134 @default.
- W115174184 cites W2027952258 @default.
- W115174184 cites W2028211844 @default.
- W115174184 cites W2028444358 @default.
- W115174184 cites W2028615902 @default.
- W115174184 cites W2031595392 @default.
- W115174184 cites W2032022374 @default.
- W115174184 cites W2032161105 @default.
- W115174184 cites W2032689093 @default.
- W115174184 cites W2033689469 @default.
- W115174184 cites W2036155956 @default.
- W115174184 cites W2036173506 @default.
- W115174184 cites W2038201387 @default.
- W115174184 cites W2039141364 @default.
- W115174184 cites W2039986849 @default.
- W115174184 cites W2041921791 @default.
- W115174184 cites W2042107934 @default.
- W115174184 cites W2042890253 @default.
- W115174184 cites W2043432548 @default.
- W115174184 cites W2045111884 @default.
- W115174184 cites W2045191357 @default.