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- W115498753 abstract "Several publications brought to light the crucial impact of CYP2C9 and more recently VKORC1 genotypes to predict dose anticoagulant requirement and thus to prevent frequent complications (including bleeding). We reported that CYP2C9 and VKORC1 genetic variations account for 50% of the drug response variability after acenocoumarol intake and showed that haplotypic study of VKORC1 was not more informative than a single SNP, corresponding to the –1639G>A promoter variation. New dosing algorithms should incorporate a single SNP (–1639G>A) and be assessed rapidly in prospective studies to help clinical settings to individualize of warfarin dose. It would be of high interest for physicians to predict about 50% of the inter-individual variability of the coumarin response by the genotyping of two SNPs, CYP2C9*3 and –1639 G>A on the VKORC1 gene." @default.
- W115498753 created "2016-06-24" @default.
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- W115498753 date "2005-01-01" @default.
- W115498753 modified "2023-09-28" @default.
- W115498753 title "Pharmacogénétique des anticoagulants oraux : variations génétiques du métabolisme et de la cible pharmacologique" @default.
- W115498753 hasPublicationYear "2005" @default.
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