Matches in SemOpenAlex for { <https://semopenalex.org/work/W129391377> ?p ?o ?g. }
- W129391377 endingPage "78" @default.
- W129391377 startingPage "49" @default.
- W129391377 abstract "Our previous studies demonstrated that progesterone down regulates the occupied form of nuclear estrogen receptor (Re). Using the density shift method, we discovered that progestins stimulate the turnover of nuclear Re within 3 h of treatment, and Re synthesis is suppressed subsequently. Thus, the primary site of progestin action in down-regulating Re is the stimulation of nuclear Re turnover followed by the inhibition of Re replenishment. A major breakthrough in our understanding of how progestin controls Re turnover was made by studying nuclear acceptor sites for Re that were found to decrease markedly within 2 h of progestin treatment. These and other results indicate that progestin induces a factor called the Re regulatory factor (ReRF) which acts to block nuclear Re acceptor sites, and this in turn decreases nuclear Re retention on chromatin acceptor sites, leading to an enhanced turnover (or processing) of nuclear Re." @default.
- W129391377 created "2016-06-24" @default.
- W129391377 creator A5020139282 @default.
- W129391377 creator A5042245279 @default.
- W129391377 creator A5049042620 @default.
- W129391377 date "1987-01-01" @default.
- W129391377 modified "2023-09-27" @default.
- W129391377 title "Progesterone-Modulation of Estrogen Action: Rapid Down Regulation of Nuclear Acceptor Sites for the Estrogen Receptor" @default.
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