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- W1490452968 endingPage "270" @default.
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- W1490452968 abstract "This chapter contains sections titled: Protein Kinase Inhibitors in Anticancer Drug Development Structure-Guided Design of Small-Molecule Inhibitors of the Cyclin-Dependent Kinases Catalytic Site Inhibitors ATP Site Specificity Alternate Strategies for Inhibiting CDKs Cyclin Groove Inhibitors (CGI) Inhibition of CDK–Cyclin Association Recent Developments in the Discovery and the Development of Aurora Kinase Inhibitors Development of Aurora Kinase Inhibitors through Screening and Structure-Guided Design Aurora Kinase Inhibitors in Clinical Trials Progress in the Identification of Potent and Selective Polo-Like Kinase Inhibitors Development of Small-Molecule Inhibitors of PLK1 Kinase Activity Discovery of Benzthiazole PLK1 Inhibitors Recent Structural Studies of the Plk1 Kinase Domain Additional Small-Molecule PLK1 Inhibitors Reported The Polo-Box Domain Future Developments References" @default.
- W1490452968 created "2016-06-24" @default.
- W1490452968 creator A5018611126 @default.
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- W1490452968 creator A5070064687 @default.
- W1490452968 date "2011-02-09" @default.
- W1490452968 modified "2023-10-14" @default.
- W1490452968 title "Discovery and Design of Protein Kinase Inhibitors: Targeting the Cell Cycle in Oncology" @default.
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