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- W1557551390 abstract "Abstract This chapter will address recent developments in the treatment of migraine. The recent promising clinical trials using a new antimigraine medication, BIBN4096BS, heralds the advent of a new generation of therapeutics. BIBN4096BS targets the receptor for the neuropeptide calcitonin gene–related peptide (CGRP), which appears to play a causal role in migraine pain. We will discuss the rationale and therapeutic implications of modulating CGRP, including its potential for acting at multiple sites in the trigeminovasculature. We will then discuss the currently used acute and preventative pharmacological treatments. Of particular interest is the increasing evidence that antiepileptic drugs may be an effective prophylactic treatment for migraine. Future strategies to selectively downregulate CGRP synthesis and the potential use of migraine drugs for other forms of trigeminal‐mediated pain, such as temporomandibular disorder and trigeminal neuralgia, will be explored." @default.
- W1557551390 created "2016-06-24" @default.
- W1557551390 creator A5000449514 @default.
- W1557551390 creator A5071785183 @default.
- W1557551390 date "2007-03-02" @default.
- W1557551390 modified "2023-10-13" @default.
- W1557551390 title "Advent of a New Generation of Antimigraine Medications" @default.
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