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- W156547202 endingPage "165" @default.
- W156547202 startingPage "103" @default.
- W156547202 abstract "An overview is presented on progress made in research on 5-HT1A receptors and their ligands since their discovery in 1983. Molecular biology has offered new tools, for example cloned 5-HT1A receptors, their mutants and chimeras to study structure and function. Many compounds, belonging to different chemical classes, display high affinity and selectivity for 5-HT1A receptors. The majority of these compounds are agonists or partial agonists, full antagonists are still scarce. Agonists and partial agonists are active in various animal models of anxiety and depression. Partial receptor agonists have been proven to be effective in general anxiety disorder and depression in man. Potential therapeutic applications for 5-HT1A receptor antagonists are evaluated, for example, in cognition disorders." @default.
- W156547202 created "2016-06-24" @default.
- W156547202 creator A5026623910 @default.
- W156547202 creator A5036713777 @default.
- W156547202 creator A5050359619 @default.
- W156547202 date "1999-01-01" @default.
- W156547202 modified "2023-10-03" @default.
- W156547202 title "The 5-HT1A receptor and its ligands: structure and function" @default.
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