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- W1572311814 endingPage "191" @default.
- W1572311814 startingPage "147" @default.
- W1572311814 abstract "A key aspect of drug action is its pharmacokinetic behavior in vivo. Because drug action depends on the drug reaching the appropriate target in vivo, positron emission tomography (PET) measurement of the tissue concentrations as a function of time in human subjects has immediate relevance to pharmacotherapy. This chapter focuses on the application of PET for the evaluation of the pharmacokinetics (PK) of small molecular weight drugs in human subjects. PET is recommended as a unique tool for comparison of aerosol drug delivery devices that deliver drugs to pulmonary tissue via oral inhalation or nasal spray. More detailed intelligence regarding the mechanism of action or the metabolism of radioactive drugs can be determined, which potentially means that the radiolabeled drug may be employed as a biomarker for noninvasive evaluation of its molecular target." @default.
- W1572311814 created "2016-06-24" @default.
- W1572311814 creator A5029519704 @default.
- W1572311814 creator A5044412006 @default.
- W1572311814 date "2013-09-20" @default.
- W1572311814 modified "2023-09-23" @default.
- W1572311814 title "PET IMAGING OF THE PHARMACOKINETICS OF SMALL MOLECULAR-WEIGHT DRUGS" @default.
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