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- W1584617434 abstract "Polymer Therapeutics can be considered among the first and most successful polymeric nanomedicines and comprises a variety of complex macromolecular systems, whose common feature is the presence of a rationally designed covalent chemical bond between a water-soluble polymeric carrier and the bioactive molecule(s). Polymer–drug conjugate concept was born with polymer chemistry adaptation for drug conjugation developed by H. Ringsdorf in 1975. Drug conjugation limits uptake to the endocytic route, favoring lysosomotropic delivery with subsequent transfer of drug out of the lysosomal compartment, providing the opportunity to bypass mechanisms of drug resistance associated with membrane efflux pumps. Involving polymer therapeutics, but not as the main actors, entails cell-based therapy transport. Batrakova et al. have developed a polyethyleneimine– poly(ethylene glycol) (PEI-PEG) complexed nanozyme loaded into bone-marrow derived monocytes (BMM) for Parkinson's disease (PD) treatment. This system was able to attenuate oxidative stress due to sustained release of the antioxidant enzyme." @default.
- W1584617434 created "2016-06-24" @default.
- W1584617434 creator A5037891181 @default.
- W1584617434 creator A5078350395 @default.
- W1584617434 creator A5083919487 @default.
- W1584617434 date "2014-10-24" @default.
- W1584617434 modified "2023-10-14" @default.
- W1584617434 title "Polymer Therapeutics as Nano‐Sized Medicines for Tissue Regeneration and Repair" @default.
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