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- W159457007 abstract "The antinociceptive and analgesic effects of muscarinic receptor ligands in human and nonhuman species have been evident for more than half a century. In this review, we describe the current understanding of the roles of different muscarinic subtypes in pain modulation and their mechanism of action along the pain signaling pathway, including peripheral nociception, spinal cord pain processing, and supraspinal analgesia. Extensive preclinical and clinical validation of these mechanisms points to the development of selective muscarinic agonists as one of the most exciting and promising avenues toward novel pain medications." @default.
- W159457007 created "2016-06-24" @default.
- W159457007 creator A5030750777 @default.
- W159457007 creator A5066816769 @default.
- W159457007 date "2011-11-03" @default.
- W159457007 modified "2023-10-06" @default.
- W159457007 title "Muscarinic Pain Pharmacology: Realizing the Promise of Novel Analgesics by Overcoming Old Challenges" @default.
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