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- W1604642011 abstract "Cytochrome P450 enzymes (CYPs) are active in the metabolism of wide variety of xenobiotics. The investigation of the contributions of human CYPs in pesticides metabolism, especially insecticides, is still growing. One of the background tools to facilitate this task is by sorting the contribution of each human CYP isoform in the metabolism of pesticides. This paper attempts to provide a comprehensive literature survey on the role of human hepatic CYPs such as human CYP1A1, CYP1A2, CYP2A6, CYP2B6, CYP2C8, CYP2C9, CYP2C19, CYP2D6, CYP2E1, CYP3A4, CYP3A5 and CYP3A7 in pesticides biotransformation in vitro as well as to sort the reactions mediated. Based on relevant publications identified by searching databases from 1995 through 2011, more than 400 metabolic reactions were reported to be mediated at least in part by human CYPs in vitro. Some information on older papers was obtained from previous literature surveys compiled by Hodgson 2001 & 2003. Finally, we give brief insight into potential modulations and consequences of human CYP genes – pesticides interactions." @default.
- W1604642011 created "2016-06-24" @default.
- W1604642011 creator A5014446196 @default.
- W1604642011 creator A5020947235 @default.
- W1604642011 creator A5028225786 @default.
- W1604642011 creator A5044013990 @default.
- W1604642011 creator A5062146319 @default.
- W1604642011 date "2012-01-05" @default.
- W1604642011 modified "2023-10-14" @default.
- W1604642011 title "Metabolism of Pesticides by Human Cytochrome P450 Enzymes In Vitro – A Survey" @default.
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