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- W1655239155 endingPage "128" @default.
- W1655239155 startingPage "95" @default.
- W1655239155 abstract "The endocannabinoids anandamide and 2-arachidonoylglycerol are metabolised by both hydrolytic enzymes (primarily fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MGL)) and oxygenating enzymes (e.g. cyclooxygenase-2, COX-2). In the present article, the in vivo data for compounds inhibiting endocannabinoid metabolism have been reviewed, focussing on inflammation and pain. Potential reasons for the failure of an FAAH inhibitor in a clinical trial in patients with osteoarthritic pain are discussed. It is concluded that there is a continued potential for compounds inhibiting endocannabinoid metabolism in terms of drug development, but that it is wise not to be unrealistic in terms of expectations of success." @default.
- W1655239155 created "2016-06-24" @default.
- W1655239155 creator A5068761485 @default.
- W1655239155 date "2015-01-01" @default.
- W1655239155 modified "2023-10-05" @default.
- W1655239155 title "The Potential of Inhibitors of Endocannabinoid Metabolism for Drug Development: A Critical Review" @default.
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