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- W167499259 abstract "This paper highlights the importance of lipid-based colloidal carriers and their pharmaceutical implications in the delivery of peptides and proteins for oral and parenteral administration. There are several examples of biomacromolecules used nowadays in the therapeutics, which are promising candidates to be delivered by means of liposomes and lipid nanoparticles, such as solid lipid nanoparticles (SLN) and nanostructured lipid carriers (NLC). Several production procedures can be applied to achieve a high association efficiency between the bioactives and the carrier, depending on the physicochemical properties of both, as well as on the production procedure applied. Generally, this can lead to improved bioavailability, or in case of oral administration a more consistent temporal profile of absorption from the gastrointestinal tract. Advantages and drawbacks of such colloidal carriers are also pointed out. This article describes strategies used for formulation of peptides and proteins, methods used for assessment of association efficiency and practical considerations regarding the toxicological concerns." @default.
- W167499259 created "2016-06-24" @default.
- W167499259 creator A5041458969 @default.
- W167499259 creator A5041950062 @default.
- W167499259 creator A5056910248 @default.
- W167499259 creator A5090966832 @default.
- W167499259 date "2007-01-01" @default.
- W167499259 modified "2023-09-29" @default.
- W167499259 title "Lipid-based colloidal carriers for peptide and protein delivery--liposomes versus lipid nanoparticles." @default.
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