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- W171773225 endingPage "233" @default.
- W171773225 startingPage "201" @default.
- W171773225 abstract "The liver is the major organ responsible for the elimination of endogenous and exogenous compounds via metabolism and/or excretion. Hepatocytes, the predominant cell type in the liver, are polarized cells with discrete basolateral and apical membranes. In this chapter, localization and function of hepatic transport proteins responsible for hepatobiliary drug disposition in humans are introduced. Hepatic transport proteins on the basolateral membrane mediate influx of compounds from sinusoidal blood into hepatocytes (i.e., NTCP, OATPs, OATs, OCTs) or efflux from hepatocytes back to sinusoidal blood (i.e., MRP3-6, OSTα/β). Canalicular transport proteins such as BSEP, MDR3, P-gp, BCRP, MRP2, and MATE1 are responsible for biliary excretion of compounds. Furthermore, in vitro (i.e., membrane vesicles, transfected cell systems, hepatocytes, isolated perfused liver) and in vivo (i.e., biliary excretion studies, hepatobiliary imaging techniques) model systems and methods that are used to investigate hepatic transport proteins are discussed, and their applications, advantages, and disadvantages are considered." @default.
- W171773225 created "2016-06-24" @default.
- W171773225 creator A5028745424 @default.
- W171773225 creator A5059675924 @default.
- W171773225 creator A5090830617 @default.
- W171773225 date "2013-01-01" @default.
- W171773225 modified "2023-10-15" @default.
- W171773225 title "Analysis of Hepatic Transport Proteins" @default.
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