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- W1723979094 abstract "Apoptosis is a mode of programmed cell death in multicellular organisms and plays a central role in controlling embryonic development, growth and differentiation and monitoring the induction of tumor cell death through anticancer therapy. Since the most effective chemotherapeutics rely on apoptosis, imaging apoptotic processes can be an invaluable tool to monitor therapeutic intervention and discover new drugs modulating apoptosis. The most attractive target for developing specific apoptosis imaging probes is caspases, crucial mediators of apoptosis. Up to now, various optical imaging strategies for apoptosis have been developed as an easy and economical modality. However, current optical applications are limited by poor sensitivity and specificity. A subset of molecular imaging contrast agents known as activatable or smart molecular probes allow for very high signal-to-background ratios compared to conventional targeted contrast agents and open up the possibility of imaging intracellular targets. In this review, we will discuss the unique design strategies and applications of activatable probes recently developed for fluorescence and bioluminescence imaging of caspase activity." @default.
- W1723979094 created "2016-06-24" @default.
- W1723979094 creator A5018249388 @default.
- W1723979094 creator A5028983150 @default.
- W1723979094 creator A5044694575 @default.
- W1723979094 date "2011-08-01" @default.
- W1723979094 modified "2023-09-23" @default.
- W1723979094 title "Design of smart probes for optical imaging of apoptosis." @default.
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- W1723979094 hasPubMedCentralId "https://www.ncbi.nlm.nih.gov/pmc/articles/3327302" @default.
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