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- W1806341467 endingPage "27" @default.
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- W1806341467 abstract "This chapter focuses on the role of adenosine triphosphate (ATP) and its metabolites as potent extracellular agents. In 1972, ATP was proposed as the transmitter responsible for nonadrenergic, noncholinergic transmission in the gut and bladder and the term “purinergic” was introduced. ATP is recognized for its important intracellular roles in many biochemical processes and is unlikely to be utilized as an extracellular messenger, although powerful extracellular enzymes involved in its breakdown are known to be present. Implicit in the concept of purinergic neurotransmission is the existence of postjunctional purinergic receptors and the potent actions of extracellular ATP on many different cell types also implicate membrane receptors. The purinergic signaling is a primitive system involved in many non-neuronal and neuronal mechanisms, including exocrine and endocrine secretion, immune responses, inflammation, pain, platelet aggregation, and endothelial-mediated vasodilatation. An increasing number of pathophysiological roles for purinoceptors are emerging, some of which have therapeutic potential. ATP stimulates pancreatic insulin release through a glucose-dependent, P2Y receptor-mediated mechanism and also modulates insulin secretion by interactions with ATP-sensitive potassium channels in islet β cells." @default.
- W1806341467 created "2016-06-24" @default.
- W1806341467 creator A5058369958 @default.
- W1806341467 date "2003-01-01" @default.
- W1806341467 modified "2023-10-17" @default.
- W1806341467 title "Introduction: ATP and Its Metabolites as Potent Extracellular Agents" @default.
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