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- W1818981862 endingPage "42" @default.
- W1818981862 startingPage "25" @default.
- W1818981862 abstract "This chapter discusses the biology and medicinal chemistry of 5-HT5A, 5-HT6 and 5-HT7 receptors. The cloning of the 5-HT5, 5-HT6 and 5-HT7 receptors has led to an increased research towards the development of selective agonists and antagonists. For example, the identification of the selective 5-HT5A antagonist 1 should provide much needed insight into the role of the 5-HT5A receptor in CNS-mediated processes. The variety and number of 5-HT6 agonists and antagonists in clinical development for obesity or cognitive disorders is representative of a large research effort from numerous pharmaceutical and academic laboratories. While there is no 5-HT7 antagonist or agonist reported to be in clinical development, the diversity of structures reported for this receptor indicates continued interest in the development of selective 5-HT7 receptor ligands with suitable drug-like properties for pre-clinical validation." @default.
- W1818981862 created "2016-06-24" @default.
- W1818981862 creator A5038074049 @default.
- W1818981862 creator A5039403483 @default.
- W1818981862 creator A5077947590 @default.
- W1818981862 date "2008-01-01" @default.
- W1818981862 modified "2023-10-17" @default.
- W1818981862 title "Recent Advances on the 5-HT5A, 5-HT6 and 5-HT7 Receptors" @default.
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