Matches in SemOpenAlex for { <https://semopenalex.org/work/W19199159> ?p ?o ?g. }
Showing items 1 to 81 of
81
with 100 items per page.
- W19199159 endingPage "3" @default.
- W19199159 startingPage "80" @default.
- W19199159 abstract "Idarubicin exhibits features rendering this drug unique among anthracyclines. The higher lipophilicity leads to faster accumulation in the nuclei, superior DNA-binding capacity and consequently greater cytotoxicity compared to daunorubicin. A major advantage over this reference drug is its ability to overcome MDR at least partially. Its major metabolite idarubicinol is as active as the parent compound and crosses the blood-brain barrier. Furthermore, idarubicin can be administered orally reaching sufficient plasma levels. Compared to other anthracyclines, the risk of cardiotoxicity as the main side effect for this group of drugs is reduced with idarubicin, when administered in a therapeutical dose. Thus, IDA has become an important drug in the treatment of acute leukemias and its potency in lymphomas, plasmocytomas and other solid tumors such as breast cancer is currently under investigation in several clinical studies." @default.
- W19199159 created "2016-06-24" @default.
- W19199159 creator A5006165963 @default.
- W19199159 creator A5057387418 @default.
- W19199159 creator A5064132655 @default.
- W19199159 creator A5084791226 @default.
- W19199159 date "1997-02-01" @default.
- W19199159 modified "2023-10-16" @default.
- W19199159 title "Idarubicin: a brief overview on pharmacology and clinical use." @default.
- W19199159 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/9147715" @default.
- W19199159 hasPublicationYear "1997" @default.
- W19199159 type Work @default.
- W19199159 sameAs 19199159 @default.
- W19199159 citedByCount "20" @default.
- W19199159 countsByYear W191991592014 @default.
- W19199159 countsByYear W191991592015 @default.
- W19199159 countsByYear W191991592016 @default.
- W19199159 crossrefType "journal-article" @default.
- W19199159 hasAuthorship W19199159A5006165963 @default.
- W19199159 hasAuthorship W19199159A5057387418 @default.
- W19199159 hasAuthorship W19199159A5064132655 @default.
- W19199159 hasAuthorship W19199159A5084791226 @default.
- W19199159 hasConcept C112705442 @default.
- W19199159 hasConcept C121608353 @default.
- W19199159 hasConcept C126322002 @default.
- W19199159 hasConcept C149151106 @default.
- W19199159 hasConcept C185592680 @default.
- W19199159 hasConcept C202751555 @default.
- W19199159 hasConcept C2776694085 @default.
- W19199159 hasConcept C2776802502 @default.
- W19199159 hasConcept C2777477808 @default.
- W19199159 hasConcept C2778233292 @default.
- W19199159 hasConcept C2779117419 @default.
- W19199159 hasConcept C2780035454 @default.
- W19199159 hasConcept C2781021840 @default.
- W19199159 hasConcept C3018657049 @default.
- W19199159 hasConcept C530470458 @default.
- W19199159 hasConcept C55493867 @default.
- W19199159 hasConcept C57992300 @default.
- W19199159 hasConcept C71924100 @default.
- W19199159 hasConcept C98274493 @default.
- W19199159 hasConceptScore W19199159C112705442 @default.
- W19199159 hasConceptScore W19199159C121608353 @default.
- W19199159 hasConceptScore W19199159C126322002 @default.
- W19199159 hasConceptScore W19199159C149151106 @default.
- W19199159 hasConceptScore W19199159C185592680 @default.
- W19199159 hasConceptScore W19199159C202751555 @default.
- W19199159 hasConceptScore W19199159C2776694085 @default.
- W19199159 hasConceptScore W19199159C2776802502 @default.
- W19199159 hasConceptScore W19199159C2777477808 @default.
- W19199159 hasConceptScore W19199159C2778233292 @default.
- W19199159 hasConceptScore W19199159C2779117419 @default.
- W19199159 hasConceptScore W19199159C2780035454 @default.
- W19199159 hasConceptScore W19199159C2781021840 @default.
- W19199159 hasConceptScore W19199159C3018657049 @default.
- W19199159 hasConceptScore W19199159C530470458 @default.
- W19199159 hasConceptScore W19199159C55493867 @default.
- W19199159 hasConceptScore W19199159C57992300 @default.
- W19199159 hasConceptScore W19199159C71924100 @default.
- W19199159 hasConceptScore W19199159C98274493 @default.
- W19199159 hasIssue "2" @default.
- W19199159 hasLocation W191991591 @default.
- W19199159 hasOpenAccess W19199159 @default.
- W19199159 hasPrimaryLocation W191991591 @default.
- W19199159 hasRelatedWork W19199159 @default.
- W19199159 hasRelatedWork W2005162843 @default.
- W19199159 hasRelatedWork W2041881020 @default.
- W19199159 hasRelatedWork W2086663675 @default.
- W19199159 hasRelatedWork W2305100815 @default.
- W19199159 hasRelatedWork W2417263408 @default.
- W19199159 hasRelatedWork W2463519831 @default.
- W19199159 hasRelatedWork W2614849848 @default.
- W19199159 hasRelatedWork W2873440957 @default.
- W19199159 hasRelatedWork W1595295580 @default.
- W19199159 hasVolume "35" @default.
- W19199159 isParatext "false" @default.
- W19199159 isRetracted "false" @default.
- W19199159 magId "19199159" @default.
- W19199159 workType "article" @default.