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- W1965280361 abstract "Bumped kinase inhibitors (BKIs) target analog-sensitive kinases, which the genomes of mammals rarely encode. Previously, we demonstrated that a BKI effectively suppressed the in vitro replication of Toxoplasma gondii, the causative pathogen of toxoplasmosis, by targeting T. gondii calcium-dependent protein kinase 1 (TgCDPK1) (Eukaryotic Cell, 9: 667-670). Here, we examined whether the BKI 1NM-PP1 reduced parasite replication in vivo. A high dose of 1NM-PP1, by intraperitoneal injection, just before the parasite inoculation effectively reduced the parasite load in the brains, livers, and lungs of T. gondii-infected mice, however, a low dose of 1NM-PP1 with oral administration didn't change the survival rates of infected mice." @default.
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- W1965280361 date "2011-01-01" @default.
- W1965280361 modified "2023-10-06" @default.
- W1965280361 title "1NM-PP1 Treatment of Mice Infected with Toxoplasma gondii" @default.
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- W1965280361 doi "https://doi.org/10.1292/jvms.11-0085" @default.
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