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- W1965774693 abstract "Agents that interfere with tubulin function have a broad anti-tumor spectrum and they represent one of the most significant classes of anticancer agents. In the past few years, several small synthetic molecules that have an indole nucleus as a core structure have been identified as tubulin inhibitors. Among these, several aroylindoles, arylthioindoles, diarylindoles and indolylglyoxyamides have shown good inhibition towards the tubulin polymerization. This article reviews the synthesis, biological activities and SARs of these main classes of indoles. Brief mention has also been made about the fused indole analogs as tubulin inhibitors." @default.
- W1965774693 created "2016-06-24" @default.
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- W1965774693 date "2012-10-01" @default.
- W1965774693 modified "2023-10-16" @default.
- W1965774693 title "Indole molecules as inhibitors of tubulin polymerization: potential new anticancer agents" @default.
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