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- W1965813305 abstract "We examined the pharmacologic effect of β-methyl-2′,6′-dimethyltyrosine-l-tetrahydroisoquinoline-3-carboxylic acid ((2S,3R)TMT-l-Tic-OH) on G protein activation in membranes prepared from Chinese Hamster Ovary cells transfected with cDNA of the human δ-opioid receptor. (2S,3R)TMT-l-Tic-OH inhibited G protein activation to 58% of basal with an EC50 of 0.72 nM as determined by [35S]GTPγS binding. These findings suggest that (2S,3R)TMT-l-Tic-OH is a highly potent inverse agonist at the human δ-opioid receptor." @default.
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- W1965813305 date "1999-09-01" @default.
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- W1965813305 title "(2S,3R)TMT-l-Tic-OH is a potent inverse agonist at the human δ-opioid receptor" @default.
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- W1965813305 doi "https://doi.org/10.1016/s0014-2999(99)00516-6" @default.
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