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- W1966336145 abstract "The effects of therapeutic concentrations of antihypertensive drugs on catechol-O-methyltransferase (COMT) and monoamine oxidase (MAO) activities in term placental explants were studied. The enzyme activities were measured in tissue fractions using radioen-zymatic techniques. At 6 h the incubation COMT activity increased significantly following exposure to verapamil and hydralazine, while exposure to alpha methyldopa caused a significant suppression of the enzyme. At 24 h exposure to hydralazine significantly suppressed the COMT activity. By 6 h the MAO activity was significantly suppressed by verapamil. MgSO4 and propranolol had no effect on the activities of COMT and MAO at 6 and 24 h. These results suggest that COMT and MAO activities in the placenta can be modulated by antihypertensive drugs and, therefore, these drugs might affect local catechol metabolism." @default.
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- W1966336145 date "1986-01-01" @default.
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- W1966336145 title "Effect of Antihypertensive Drugs on Catechol-O-Methyltransferase and Monoamine Oxidase Activity in Human Term Placental Explants" @default.
- W1966336145 doi "https://doi.org/10.1159/000298941" @default.
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