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- W1966700703 abstract "Drug design: Oxazoles and thiazoles were designed and synthesised based on previously reported ligands of the 3rd histamine receptor (H3R). The aminopropoxy-phenyl-oxazole chemotype was identified as a promising H3R inverse agonist with superior drug-like properties, good efficacy in vivo and good safety margin." @default.
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- W1966700703 date "2010-01-26" @default.
- W1966700703 modified "2023-10-17" @default.
- W1966700703 title "Phenyl-oxazoles, a New Family of Inverse Agonists at the H<sub>3</sub>Histamine Receptor" @default.
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- W1966700703 doi "https://doi.org/10.1002/cmdc.200900446" @default.
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