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- W1967316295 abstract "The inside cover picture shows a carbazole (compd 25 in the article) interacting with both P-glycoprotein (P-gp) and σ2 receptors. Through these combined activities, a futile ATP cycle is activated and reactive oxygen species (ROS) are generated. Enhanced antiproliferative effects were observed in drug-resistant over standard MCF7 cells. This phenomenon, termed collateral sensitivity, is under study in multidrug- resistant tumors, and mixed σ2 agonists/P-gp substrates are promising for their treatment. For more details, see the Full Paper by Carmen Abate et al. on p. 2026 ff." @default.
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- W1967316295 date "2013-11-29" @default.
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- W1967316295 title "Inside Cover: Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity (ChemMedChem 12/2013)" @default.
- W1967316295 doi "https://doi.org/10.1002/cmdc.201390051" @default.
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