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- W1969915718 abstract "A set of equations was applied that allows the use of racemic mixtures for the estimation of kinetic parameters in systems where the l-isomer is substrate and the d-isomer a competitive inhibitor, displaying data as double reciprocal plots. A statistical treatment was introduced that renders compatible the output of presently available programs with the specific model requirements, with few additional calculations. An example is shown with β-trypsin and its inhibition of benzozyl-d-arginine p-nitroanilide (Ki = 1.12 mM, pH 8,0, 37 °C)." @default.
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- W1969915718 date "1984-01-01" @default.
- W1969915718 modified "2023-10-18" @default.
- W1969915718 title "Competitive inhibition by the d-isomer in racemic mixtures used as substrate in kinetic studies: A simple method for data treatment" @default.
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- W1969915718 doi "https://doi.org/10.1016/0003-9861(84)90068-7" @default.
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