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- W1971294725 abstract "1. The effects of ivermectin (IVM) and milbemycin D (MMD) on cultured embryonic spinal neurons were investigated, using the whole-cell recording technique. 2. IVM and MMD caused Cl- current under voltage-clamp conditions. 3. The reversal potential of the MMD-evoked Cl- current was shifted in a positive direction when half of the external Cl- was substituted by isethionate. 4. The MMD-evoked current was inhibited by picrotoxinin and bicuculline, whereas it was enhanced by diazepam. 5. Different characteristics of desensitization were observed between the MMD- (IVM-) and muscimol-induced effects. 6. These results suggest that IVM and MMD directly activate the Cl- channel through their specific sites modulated by GABAergic drugs." @default.
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- W1971294725 date "1989-01-01" @default.
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- W1971294725 title "Macrolide compounds, ivermectin and milbemycin D, stimulate chloride channels sensitive to gabaergic drugs in cultured chick spinal neurons" @default.
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- W1971294725 doi "https://doi.org/10.1016/0742-8413(89)90017-0" @default.
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