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- W1972624770 abstract "Cathepsin S is a potential target of autoimmune disease. A series of proline derived compounds were synthesized and evaluated as cathepsin S inhibitors. We discovered potent cathepsin S inhibitors through structure–activity relationship studies of proline analogues. In particular, compound 19-(S) showed promising in vitro/vivo pharmacological activities and properties as a selective cathepsin S inhibitor." @default.
- W1972624770 created "2016-06-24" @default.
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- W1972624770 date "2013-06-01" @default.
- W1972624770 modified "2023-09-24" @default.
- W1972624770 title "Synthesis of proline analogues as potent and selective cathepsin S inhibitors" @default.
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- W1972624770 doi "https://doi.org/10.1016/j.bmcl.2013.04.023" @default.
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