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- W1974283835 abstract "Novel antibacterial fluoroquinolone agents bearing a 4-alkylidenylpiperidine 7-position substituent are active against quinolone-susceptible and quinolone-resistant gram-positive bacteria, including Streptococcus pneumoniae and MRSA. Analogs 22b, 23c, and 24 demonstrated superior in vitro and in vivo efficacy to ciprofloxacin against these cocci." @default.
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- W1974283835 date "2014-12-01" @default.
- W1974283835 modified "2023-10-18" @default.
- W1974283835 title "7-(4-Alkylidenylpiperidinyl)-quinolone bacterial topoisomerase inhibitors" @default.
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- W1974283835 doi "https://doi.org/10.1016/j.bmcl.2014.10.014" @default.
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