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- W1976366904 abstract "The disposition kinetics of difloxacin, a fluoroquinolone antibiotic, after intravenous (IV), intramuscular (IM) and subcutaneous (SC) administration were determined in sheep at a single dose of 5 mg/kg. The concentration–time data were analysed by compartmental (after IV dose) and non-compartmental pharmacokinetics method (after IV, IM and SC administration). Plasma concentrations of difloxacin were determined by high performance liquid chromatography with fluorescence detection. Steady-state volume of distribution (Vss) and clearance (Cl) of difloxacin after IV administration were 1.68 ± 0.21 L/kg and 0.21 ± 0.03 L/h kg, respectively. Following IM and SC administration difloxacin achieved maximum plasma concentration of 1.89 ± 0.55 and 1.39 ± 0.14 mg/L at 2.42 ± 1.28 and 5.33 ± 1.03 h, respectively. The absolute bioavailabilities after IM and SC routes were 99.92 ± 26.50 and 82.35 ± 25.65%, respectively. Based on these kinetic parameters, difloxacin is likely to be effective in sheep." @default.
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- W1976366904 date "2007-10-01" @default.
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- W1976366904 title "Pharmacokinetics after intravenous, intramuscular and subcutaneous administration of difloxacin in sheep" @default.
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- W1976366904 doi "https://doi.org/10.1016/j.rvsc.2007.01.005" @default.
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