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- W1977778248 abstract "Basal ganglia processing results from a balanced activation of direct and indirect striatal efferent pathways, which are controlled by dopamine D 1 and D 2 receptors, respectively. Adenosine A 2A receptors are considered novel antiparkinsonian targets, based on their selective postsynaptic localization in the indirect pathway, where they modulate D 2 receptor function. The present study provides evidence for the existence of an additional, functionally significant, segregation of A 2A receptors at the presynaptic level. Using integrated anatomical, electrophysiological, and biochemical approaches, we demonstrate that presynaptic A 2A receptors are preferentially localized in cortical glutamatergic terminals that contact striatal neurons of the direct pathway, where they exert a selective modulation of corticostriatal neurotransmission. Presynaptic striatal A 2A receptors could provide a new target for the treatment of neuropsychiatric disorders." @default.
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- W1977778248 date "2009-01-01" @default.
- W1977778248 modified "2023-10-17" @default.
- W1977778248 title "Key Modulatory Role of Presynaptic Adenosine A<sub>2A</sub>Receptors in Cortical Neurotransmission to the Striatal Direct Pathway" @default.
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- W1977778248 doi "https://doi.org/10.1100/tsw.2009.143" @default.
- W1977778248 hasPubMedCentralId "https://www.ncbi.nlm.nih.gov/pmc/articles/2871285" @default.
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