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- W1978522011 abstract "Using a high-throughput screening campaign, we identified the 4,6-bis anilino pyrimidines as inhibitors of the cyclin-dependent kinase, CDK4. Herein we describe the further chemical modification and use of X-ray crystallography to develop potent and selective in vitro inhibitors of CDK4." @default.
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- W1978522011 date "2003-09-01" @default.
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- W1978522011 title "Cyclin-dependent kinase 4 inhibitors as a treatment for cancer. Part 1: identification and optimisation of substituted 4,6-Bis anilino pyrimidines" @default.
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- W1978522011 doi "https://doi.org/10.1016/s0960-894x(03)00202-6" @default.
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