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- W1978917215 endingPage "540" @default.
- W1978917215 startingPage "520" @default.
- W1978917215 abstract "Immortality of tumour cells is strictly correlated to telomerase activity. Telomerase is overexpressed in about 85% of tumour cells and maintains telomere length contributing to cell immortalisation, whereas in somatic cells telomeres progressively shorten until cell death occurs by apoptosis. Different drugs can promote telomeric G-rich overhangs which fold into quadruplex structures that inhibit telomerase activity. Detailed studies on drug-quadruplex complexes are essential to understand quadruplex recognition and address drug design. This review will discuss the energetic aspects of quadruplex-drug interactions with a particular attention to physico-chemical methodologies. Keywords: Telomerase, telomeric DNA, G-quadruplex, G-quadruplex-drug interactions, physico-chemical techniques" @default.
- W1978917215 created "2016-06-24" @default.
- W1978917215 creator A5068253734 @default.
- W1978917215 creator A5068862723 @default.
- W1978917215 date "2007-09-01" @default.
- W1978917215 modified "2023-09-23" @default.
- W1978917215 title "Energetics of Quadruplex-Drug Recognition in Anticancer Therapy" @default.
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