Matches in SemOpenAlex for { <https://semopenalex.org/work/W1983027650> ?p ?o ?g. }
- W1983027650 endingPage "369" @default.
- W1983027650 startingPage "363" @default.
- W1983027650 abstract "1. In 64 patients undergoing coronary artery bypass grafting the effects of chronic beta 1-adrenoceptor antagonist (metoprolol, atenolol, bisoprolol) treatment on right atrial beta-adrenoceptor and muscarinic M2-receptor number and functional responsiveness were investigated. 2. The beta 1-adrenoceptor antagonists increased right atrial beta 1-adrenoceptor number, did not affect beta 2-adrenoceptor number, and decreased muscarinic M2-receptor number. 3. Concomitantly, activation of right atrial adenylate cyclase by 10 microM GTP, 10 microM isoprenaline and 1 microM forskolin was enhanced and inhibition by 100 microM carbachol was diminished. 4. On isolated, electrically driven right atria the beta 1-adrenoceptor-mediated positive inotropic effect of noradrenaline was - even with beta 1-adrenoceptor number increased - not altered, while the beta 2-adrenoceptor-mediated effect of procaterol was markedly enhanced. However, the carbachol-induced negative inotropic effect was decreased. 5. It is concluded that chronic beta 1-adrenoceptor antagonist treatment increases beta 1-adrenoceptor number and concomitantly sensitizes beta 2-adrenoceptor function, but desensitizes muscarinic M2-receptor function in the human heart." @default.
- W1983027650 created "2016-06-24" @default.
- W1983027650 creator A5003482863 @default.
- W1983027650 creator A5009800572 @default.
- W1983027650 creator A5030074177 @default.
- W1983027650 creator A5040869371 @default.
- W1983027650 creator A5045246727 @default.
- W1983027650 creator A5063355903 @default.
- W1983027650 date "1990-10-01" @default.
- W1983027650 modified "2023-10-17" @default.
- W1983027650 title "Chronic β1-adrenoceptor antagonist treatment sensitizes β2-adrenoceptors, but desensitizes M2-muscarinic receptors in the human right atrium" @default.
- W1983027650 cites W159198934 @default.
- W1983027650 cites W1775749144 @default.
- W1983027650 cites W1983649348 @default.
- W1983027650 cites W1983840966 @default.
- W1983027650 cites W1988675802 @default.
- W1983027650 cites W2003055956 @default.
- W1983027650 cites W2009310647 @default.
- W1983027650 cites W2010527717 @default.
- W1983027650 cites W2013475109 @default.
- W1983027650 cites W2022946669 @default.
- W1983027650 cites W2023675599 @default.
- W1983027650 cites W2025456951 @default.
- W1983027650 cites W2043536009 @default.
- W1983027650 cites W2044728148 @default.
- W1983027650 cites W2045384414 @default.
- W1983027650 cites W2050153950 @default.
- W1983027650 cites W2054894807 @default.
- W1983027650 cites W2055398677 @default.
- W1983027650 cites W2057451767 @default.
- W1983027650 cites W2062304838 @default.
- W1983027650 cites W2066920501 @default.
- W1983027650 cites W2067015973 @default.
- W1983027650 cites W2074192832 @default.
- W1983027650 cites W2075827507 @default.
- W1983027650 cites W2081559057 @default.
- W1983027650 cites W2088672176 @default.
- W1983027650 cites W2089959767 @default.
- W1983027650 cites W2092082950 @default.
- W1983027650 cites W2140509492 @default.
- W1983027650 cites W2146333603 @default.
- W1983027650 cites W2154329909 @default.
- W1983027650 cites W2278336196 @default.
- W1983027650 cites W2322567932 @default.
- W1983027650 cites W2339250602 @default.
- W1983027650 cites W4230304113 @default.
- W1983027650 cites W44420309 @default.
- W1983027650 doi "https://doi.org/10.1111/j.1476-5381.1990.tb12715.x" @default.
- W1983027650 hasPubMedCentralId "https://www.ncbi.nlm.nih.gov/pmc/articles/1917687" @default.
- W1983027650 hasPubMedId "https://pubmed.ncbi.nlm.nih.gov/1979509" @default.
- W1983027650 hasPublicationYear "1990" @default.
- W1983027650 type Work @default.
- W1983027650 sameAs 1983027650 @default.
- W1983027650 citedByCount "81" @default.
- W1983027650 countsByYear W19830276502012 @default.
- W1983027650 countsByYear W19830276502013 @default.
- W1983027650 countsByYear W19830276502014 @default.
- W1983027650 countsByYear W19830276502015 @default.
- W1983027650 countsByYear W19830276502018 @default.
- W1983027650 countsByYear W19830276502020 @default.
- W1983027650 countsByYear W19830276502021 @default.
- W1983027650 crossrefType "journal-article" @default.
- W1983027650 hasAuthorship W1983027650A5003482863 @default.
- W1983027650 hasAuthorship W1983027650A5009800572 @default.
- W1983027650 hasAuthorship W1983027650A5030074177 @default.
- W1983027650 hasAuthorship W1983027650A5040869371 @default.
- W1983027650 hasAuthorship W1983027650A5045246727 @default.
- W1983027650 hasAuthorship W1983027650A5063355903 @default.
- W1983027650 hasBestOaLocation W19830276501 @default.
- W1983027650 hasConcept C126322002 @default.
- W1983027650 hasConcept C134018914 @default.
- W1983027650 hasConcept C15324608 @default.
- W1983027650 hasConcept C170493617 @default.
- W1983027650 hasConcept C185592680 @default.
- W1983027650 hasConcept C24998067 @default.
- W1983027650 hasConcept C2776090920 @default.
- W1983027650 hasConcept C2776525901 @default.
- W1983027650 hasConcept C2776663762 @default.
- W1983027650 hasConcept C2776723954 @default.
- W1983027650 hasConcept C2776885963 @default.
- W1983027650 hasConcept C2778151854 @default.
- W1983027650 hasConcept C2778198053 @default.
- W1983027650 hasConcept C2778988552 @default.
- W1983027650 hasConcept C2779276759 @default.
- W1983027650 hasConcept C2779670145 @default.
- W1983027650 hasConcept C33789571 @default.
- W1983027650 hasConcept C71924100 @default.
- W1983027650 hasConcept C84393581 @default.
- W1983027650 hasConceptScore W1983027650C126322002 @default.
- W1983027650 hasConceptScore W1983027650C134018914 @default.
- W1983027650 hasConceptScore W1983027650C15324608 @default.
- W1983027650 hasConceptScore W1983027650C170493617 @default.
- W1983027650 hasConceptScore W1983027650C185592680 @default.
- W1983027650 hasConceptScore W1983027650C24998067 @default.
- W1983027650 hasConceptScore W1983027650C2776090920 @default.
- W1983027650 hasConceptScore W1983027650C2776525901 @default.
- W1983027650 hasConceptScore W1983027650C2776663762 @default.
- W1983027650 hasConceptScore W1983027650C2776723954 @default.