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- W1984734436 abstract "A series of 2-aminomethyl piperidines has been discovered as novel urotensin-II receptor antagonists. The synthesis, initial structure-activity relationships, and optimization of the initial hit that resulted in the identification of potent, cross-species active, and functional urotensin-II receptor antagonists such as 1a and 11a are described." @default.
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- W1984734436 date "2008-05-01" @default.
- W1984734436 modified "2023-09-27" @default.
- W1984734436 title "2-Aminomethyl piperidines as novel urotensin-II receptor antagonists" @default.
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- W1984734436 doi "https://doi.org/10.1016/j.bmcl.2008.03.078" @default.
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