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- W1985356444 endingPage "45" @default.
- W1985356444 startingPage "27" @default.
- W1985356444 abstract "Methods employing in vitro and in situ means can be used to gain early information regarding the potential for intestinal absorption of new chemical entities (NCEs). Physicochemical and biological approaches for evaluation of the intestinal absorption of NCEs are described in this review. Physicochemical measurements such as aqueous solubility, lipophilicity and membrane partioning form an important base for subsequent biological experiments. Biological techniques that include subcellular membrane fractions, intestinal cells, isolated tissue and organ perfusion are detailed. Several of these preparations can be utilized for transport, as well as stability indicators. While some methods are generally applicable to NCEs, others require selectivity on the part of the investigator, depending on the information desired." @default.
- W1985356444 created "2016-06-24" @default.
- W1985356444 creator A5045696947 @default.
- W1985356444 creator A5061354362 @default.
- W1985356444 creator A5073057060 @default.
- W1985356444 creator A5077342644 @default.
- W1985356444 date "1997-01-01" @default.
- W1985356444 modified "2023-10-17" @default.
- W1985356444 title "Discrimination between drug candidates using models for evaluation of intestinal absorption" @default.
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