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- W1987965251 abstract "Abstract: The effect on excitatory amino acid (EAA)-induced toxicity of two novel non-N-methyl-d-aspartate (non-NMDA) antagonists 2-amino-3-[3-(carboxymethoxy)-5-methylisoxazol-4-yl]propionic acid (AMOA) and 2-amino-3-[2-(3-hydroxy-5-methyl-isoxazol-4-yl)methyl-5-methyl-3-oxoisoxazolin-4-yl]propionic acid (AMNH) was tested in primary cultures of cerebral cortex neurons. Such cultures provide a useful model for the investigation of the toxicity of EAAs and a convenient screening system for potential neuroprotective activity of pharmacological agents. It was demonstrated that AMNH and AMOA abolished neurotoxicity induced by kainic acid with IC50 values of 62 ± 10 and 120 ± 19 μM, respectively. No effect on neuronal damage induced by NMDA or AMPA could be detected." @default.
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- W1987965251 date "1990-11-01" @default.
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- W1987965251 title "Novel Glutamate Receptor Antagonists Selectively Protect Against Kainic Acid Neurotoxicity in Cultured Cerebral Cortex Neurons" @default.
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- W1987965251 doi "https://doi.org/10.1111/j.1471-4159.1990.tb04976.x" @default.
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