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- W1988227670 endingPage "1885" @default.
- W1988227670 startingPage "1875" @default.
- W1988227670 abstract "Nuclear factor-erythroid 2 p45-related factor 2 (NRF2, also known as Nfe2l2) plays a critical role in regulating cellular defense against electrophilic and oxidative stress by activating the expression of an array of antioxidant response element-dependent genes. On one hand, NRF2 activators have been used in clinical trials for cancer prevention and the treatment of diseases associated with oxidative stress; on the other hand, constitutive activation of NRF2 in many types of tumors contributes to the survival and growth of cancer cells, as well as resistance to anticancer therapy. In this review, we provide an overview of the NRF2 signaling pathway and discuss its role in carcinogenesis. We also introduce the inhibition of NRF2 by nuclear receptors. Further, we address the biological significance of regulation of the NRF2 signaling pathway by nuclear receptors in health and disease. Finally, we discuss the possible impact of NRF2 inhibition by nuclear receptors on cancer therapy." @default.
- W1988227670 created "2016-06-24" @default.
- W1988227670 creator A5038339399 @default.
- W1988227670 creator A5057134186 @default.
- W1988227670 creator A5068397352 @default.
- W1988227670 creator A5087124601 @default.
- W1988227670 date "2014-09-01" @default.
- W1988227670 modified "2023-10-16" @default.
- W1988227670 title "Modulation of NRF2 signaling pathway by nuclear receptors: Implications for cancer" @default.
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