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- W1988522068 abstract "Constitutive activation of the EPO/JAK2 signaling cascade has recently been implicated in a variety of myeloproliferative disorders including polycythemia vera, essential thrombocythemia and myelofibrosis. In an effort to uncover therapeutic potential of blocking the EPO/JAK2 signaling cascade, we sought to discover selective inhibitors that block the kinase activity of JAK2. Herein, we describe the discovery and structure based optimization of a novel series of 2-amino-pyrazolo[1,5-a]pyrimidines that exhibit potent inhibition of JAK2." @default.
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- W1988522068 date "2009-12-01" @default.
- W1988522068 modified "2023-10-14" @default.
- W1988522068 title "2-Aminopyrazolo[1,5-a]pyrimidines as potent and selective inhibitors of JAK2" @default.
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- W1988522068 doi "https://doi.org/10.1016/j.bmcl.2009.10.053" @default.
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