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- W1990264609 abstract "The effectiveness of several detergents and salts in solubilizing the muscarinic acetylcholine receptor (identified by its atropine-sensitive [3H]3-quinuclidinyl benzilate (QNB) binding) from bovine striatal membranes is reported. The highest density of receptor is obtained by extraction with 1% digitonin-0.1 mM EDTA. Although the total solubilized muscarinic receptors (sites/ml) are increased and the nonspecific binding is decreased when 1 M NaCl is included in this extraction medium, the receptor density (sites/mg protein) is lower. The solubilized receptors have the same specific QNB binding affinity, and sensitivity to a variety of drugs, as the membrane-bound muscarinic receptors." @default.
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- W1990264609 date "1978-10-01" @default.
- W1990264609 modified "2023-09-23" @default.
- W1990264609 title "Solubilization of muscarinic acetylcholine receptors of bovine brain" @default.
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- W1990264609 doi "https://doi.org/10.1016/0024-3205(78)90397-1" @default.
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