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- W1990696688 abstract "The design and synthesis of a novel series of potent gamma secretase modulators is described. Exploration of various spacer groups between the triazole ring and the aromatic appendix in 2 has led to anilinotriazole 28, which combined high in vitro and in vivo potency with an acceptable drug-like profile." @default.
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- W1990696688 date "2014-12-01" @default.
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- W1990696688 title "Anilinotriazoles as potent gamma secretase modulators" @default.
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- W1990696688 doi "https://doi.org/10.1016/j.bmcl.2014.10.024" @default.
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