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- W1992826986 abstract "Le rein joue un rôle central dans le métabolisme du glucose et la régulation de la glycémie. Le cotransporteur sodium glucose de type 2 (SGLT2) rénal a un rôle clé dans le transport actif du glucose en régulant la réabsorption rénale du glucose et représente donc une cible pharmacologique potentielle pour le traitement du diabète. Les effets des inhibiteurs du SGLT2 dans les modèles animaux, ainsi que les données actuellement disponibles des études cliniques de phase 2 conduites, en administration orale, chez des patients ayant un diabète de type 2 avec des inhibiteurs sélectifs de SGLT2 sont présentées et discutées. The kidney has an important role in glucose metabolism and regulation. The renal sodium glucose co-transporter 2 (SGLT2) has a key role in the active transport of glucose by determining renal glucose reabsorption, thus representing a potential target for pharmacological diabetes treatment. Effects of SGLT2 inhibitors in various animal models, as well as currently available phase 2 clinical results with oral selective SGLT2 inhibitors in type 2 diabetic patients are presented and discussed." @default.
- W1992826986 created "2016-06-24" @default.
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- W1992826986 date "2009-09-01" @default.
- W1992826986 modified "2023-09-25" @default.
- W1992826986 title "Inhibiteurs du cotransporteur sodium-glucose de type 2 (SGLT2) : une nouvelle approche thérapeutique pour le diabète de type 2 ?" @default.
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- W1992826986 doi "https://doi.org/10.1016/s1957-2557(09)72401-0" @default.
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