Matches in SemOpenAlex for { <https://semopenalex.org/work/W1992907077> ?p ?o ?g. }
- W1992907077 endingPage "102" @default.
- W1992907077 startingPage "92" @default.
- W1992907077 abstract "Central nervous system (CNS) drug delivery remains a major challenge, despite extensive efforts that have been made to develop novel strategies to overcome obstacles. Prodrugs are bioreversible derivatives of drug molecules that must undergo an enzymatic and/or chemical transformation in vivo to release the active parent drug, which subsequently exerts the desired pharmacological effect. In both drug discovery and drug development, prodrugs have become an established tool for improving physicochemical, biopharmaceutical or pharmacokinetic properties of pharmacologically active agents that overcome barriers to a drug's usefulness. This review provides insight into various prodrug strategies explored to date for CNS drug delivery, including lipophilic prodrugs, carrier- and receptor-mediated prodrug delivery systems, and gene-directed enzyme prodrug therapy." @default.
- W1992907077 created "2016-06-24" @default.
- W1992907077 creator A5030482084 @default.
- W1992907077 creator A5033453163 @default.
- W1992907077 creator A5051447344 @default.
- W1992907077 creator A5063971478 @default.
- W1992907077 date "2008-02-05" @default.
- W1992907077 modified "2023-10-12" @default.
- W1992907077 title "Prodrug Approaches for CNS Delivery" @default.
- W1992907077 cites W100906034 @default.
- W1992907077 cites W111781460 @default.
- W1992907077 cites W113805164 @default.
- W1992907077 cites W127754072 @default.
- W1992907077 cites W1513790751 @default.
- W1992907077 cites W1541915068 @default.
- W1992907077 cites W1574468119 @default.
- W1992907077 cites W1964598686 @default.
- W1992907077 cites W1966538775 @default.
- W1992907077 cites W1969899703 @default.
- W1992907077 cites W1970263371 @default.
- W1992907077 cites W1973308376 @default.
- W1992907077 cites W1973544766 @default.
- W1992907077 cites W1975947373 @default.
- W1992907077 cites W1976678915 @default.
- W1992907077 cites W1977643218 @default.
- W1992907077 cites W1979657535 @default.
- W1992907077 cites W1984399394 @default.
- W1992907077 cites W1985944040 @default.
- W1992907077 cites W1986144289 @default.
- W1992907077 cites W1992983740 @default.
- W1992907077 cites W1994532346 @default.
- W1992907077 cites W1996499842 @default.
- W1992907077 cites W2001097099 @default.
- W1992907077 cites W2006670903 @default.
- W1992907077 cites W2011225701 @default.
- W1992907077 cites W2015625626 @default.
- W1992907077 cites W2017952116 @default.
- W1992907077 cites W2018777412 @default.
- W1992907077 cites W2019243633 @default.
- W1992907077 cites W2020291065 @default.
- W1992907077 cites W2023410591 @default.
- W1992907077 cites W2028441136 @default.
- W1992907077 cites W2032973723 @default.
- W1992907077 cites W2035966615 @default.
- W1992907077 cites W2038182972 @default.
- W1992907077 cites W2038629387 @default.
- W1992907077 cites W2040169414 @default.
- W1992907077 cites W2041140779 @default.
- W1992907077 cites W2043355351 @default.
- W1992907077 cites W2044446715 @default.
- W1992907077 cites W2046826638 @default.
- W1992907077 cites W2048291054 @default.
- W1992907077 cites W2049309316 @default.
- W1992907077 cites W2050502325 @default.
- W1992907077 cites W2051188685 @default.
- W1992907077 cites W2054140553 @default.
- W1992907077 cites W2055137287 @default.
- W1992907077 cites W2055233461 @default.
- W1992907077 cites W2056257486 @default.
- W1992907077 cites W2059183805 @default.
- W1992907077 cites W2060432355 @default.
- W1992907077 cites W2062421366 @default.
- W1992907077 cites W2064169769 @default.
- W1992907077 cites W2064873536 @default.
- W1992907077 cites W2065318944 @default.
- W1992907077 cites W2065452150 @default.
- W1992907077 cites W2065734111 @default.
- W1992907077 cites W2074919840 @default.
- W1992907077 cites W2077182842 @default.
- W1992907077 cites W2077643551 @default.
- W1992907077 cites W2080911783 @default.
- W1992907077 cites W2081959205 @default.
- W1992907077 cites W2083274261 @default.
- W1992907077 cites W2084338973 @default.
- W1992907077 cites W2087666006 @default.
- W1992907077 cites W2092108048 @default.
- W1992907077 cites W2095512576 @default.
- W1992907077 cites W2101099825 @default.
- W1992907077 cites W2101193630 @default.
- W1992907077 cites W2104290477 @default.
- W1992907077 cites W2113634953 @default.
- W1992907077 cites W2117265627 @default.
- W1992907077 cites W2122195853 @default.
- W1992907077 cites W2123424839 @default.
- W1992907077 cites W2126349589 @default.
- W1992907077 cites W2128890618 @default.
- W1992907077 cites W2130695898 @default.
- W1992907077 cites W2139732917 @default.
- W1992907077 cites W2148756948 @default.
- W1992907077 cites W2151199853 @default.
- W1992907077 cites W2151440675 @default.
- W1992907077 cites W2152353759 @default.
- W1992907077 cites W2161343130 @default.
- W1992907077 cites W2164752182 @default.
- W1992907077 cites W2169879202 @default.
- W1992907077 cites W2172477250 @default.
- W1992907077 cites W2331944802 @default.
- W1992907077 cites W2341202044 @default.